| Cathepsin B: Active site mapping with peptidic substrates and inhibitors J Schmitz, E Gilberg, R Löser, J Bajorath, U Bartz, M Gütschow Bioorganic & medicinal chemistry 27 (1), 1-15, 2019 | 58 | 2019 |
| A Coumarin‐Labeled Vinyl Sulfone as Tripeptidomimetic Activity‐Based Probe for Cysteine Cathepsins MD Mertens, J Schmitz, M Horn, N Furtmann, J Bajorath, M Mareš, ... ChemBioChem 15 (7), 955-959, 2014 | 57 | 2014 |
| Evaluation of dipeptide nitriles as inhibitors of rhodesain, a major cysteine protease of Trypanosoma brucei T Schirmeister, J Schmitz, S Jung, T Schmenger, RL Krauth-Siegel, ... Bioorganic & Medicinal Chemistry Letters 27 (1), 45-50, 2017 | 45 | 2017 |
| Cathepsin B inhibitors: combining dipeptide nitriles with an occluding loop recognition element by click chemistry J Schmitz, T Li, U Bartz, M Gütschow ACS Medicinal Chemistry Letters 7 (3), 211-216, 2016 | 32 | 2016 |
| Design, characterization and cellular uptake studies of fluorescence-labeled prototypic cathepsin inhibitors F Kohl, J Schmitz, N Furtmann, AC Schulz-Fincke, MD Mertens, J Küppers, ... Organic & Biomolecular Chemistry 13 (41), 10310-10323, 2015 | 26 | 2015 |
| Selective nitrile inhibitors to modulate the proteolytic synergism of cathepsins S and F M Frizler, J Schmitz, AC Schulz-Fincke, M Gütschow Journal of Medicinal Chemistry 55 (12), 5982-5986, 2012 | 19 | 2012 |
| 3-Cyano-3-aza-β-amino acid derivatives as inhibitors of human cysteine cathepsins J Schmitz, AM Beckmann, A Dudic, T Li, R Sellier, U Bartz, M Gütschow ACS Medicinal Chemistry Letters 5 (10), 1076-1081, 2014 | 17 | 2014 |
| An Access to Aza-Freidinger Lactams and E-Locked Analogs PA Ottersbach, J Schmitz, G Schnakenburg, M Gütschow Organic letters 15 (3), 448-451, 2013 | 14 | 2013 |
| 3, 5, 5-Trisubstituted hydantoins from activated (benzyloxycarbonylamino) malonic acids L Hroch, M Hrušková, J Schmitz, G Schnakenburg, M Guetschow Synthesis 44 (12), 1907-1914, 2012 | 12 | 2012 |
| Synthesis and kinetic evaluation of ethyl acrylate and vinyl sulfone derived inhibitors for human cysteine cathepsins C Breuer, C Lemke, J Schmitz, U Bartz, M Gütschow Bioorganic & Medicinal Chemistry Letters 28 (11), 2008-2012, 2018 | 8 | 2018 |
| Active site mapping of human cathepsin F with dipeptide nitrile inhibitors J Schmitz, N Furtmann, M Ponert, M Frizler, R Löser, U Bartz, J Bajorath, ... ChemMedChem 10 (8), 1365-1377, 2015 | 5 | 2015 |
| Transformation of the carboxyl group of an amino acid to variously substituted imidazoles through a Davidson-type heterocyclization J Kueppers, M Hympanova, T Keuler, AJ Schneider, G Schnakenburg, ... Synthesis 51 (09), 1961-1968, 2019 | 1 | 2019 |
| Active Site Mapping of Human Cathepsin F with Dipeptide Nitrile Inhibitors J Schmitz, N Furtmann, M Ponert, U Bartz, J Bajorath, M Gütschow Drug Discovery and Therapy World Congress 2015, 182, 2016 | | 2016 |
| Synthesis and biological evaluation of nitrile-based peptiomimetic inhibitors fore cysteine cathepsins J Schmitz | | 2016 |
