Filtering promiscuous compounds in early drug discovery: is it a good idea? MR Senger, CAM Fraga, RF Dantas, FP Silva Jr Drug Discovery Today 21 (6), 868-872, 2016 | 96 | 2016 |
ATP and ADP hydrolysis in brain membranes of zebrafish (Danio rerio) EP Rico, MR Senger, M da Graça Fauth, RD Dias, MR Bogo, CD Bonan Life Sciences 73 (16), 2071-2082, 2003 | 94 | 2003 |
Methanol alters ecto-nucleotidases and acetylcholinesterase in zebrafish brain EP Rico, DB Rosemberg, MR Senger, M de Bem Arizi, GF Bernardi, ... Neurotoxicology and Teratology 28 (4), 489-496, 2006 | 92 | 2006 |
Ecto-5′-nucleotidase activity in brain membranes of zebrafish (Danio rerio) MR Senger, EP Rico, RD Dias, MR Bogo, CD Bonan Comparative Biochemistry and Physiology Part B: Biochemistry and Molecular …, 2004 | 84 | 2004 |
Exposure to Hg2+ and Pb2+ changes NTPDase and ecto-5′-nucleotidase activities in central nervous system of zebrafish (Danio rerio) MR Senger, EP Rico, M de Bem Arizi, APG Frazzon, RD Dias, MR Bogo, ... Toxicology 226 (2-3), 229-237, 2006 | 81 | 2006 |
Aluminum exposure alters behavioral parameters and increases acetylcholinesterase activity in zebrafish (Danio rerio) brain MR Senger, KJ Seibt, GC Ghisleni, RD Dias, MR Bogo, CD Bonan Cell biology and toxicology 27, 199-205, 2011 | 80 | 2011 |
Discovery of new anti-schistosomal hits by integration of QSAR-based virtual screening and high content screening BJ Neves, RF Dantas, MR Senger, CC Melo-Filho, WCG Valente, ... Journal of medicinal chemistry 59 (15), 7075-7088, 2016 | 77 | 2016 |
1-Phenyl-1H-and 2-phenyl-2H-1, 2, 3-triazol derivatives: Design, synthesis and inhibitory effect on alpha-glycosidases D Gonzaga, MR Senger, FC Da Silva, VF Ferreira, FP Silva-Jr European Journal of Medicinal Chemistry 74, 461-476, 2014 | 72 | 2014 |
In vitro effect of zinc and cadmium on acetylcholinesterase and ectonucleotidase activities in zebrafish (Danio rerio) brain MR Senger, DB Rosemberg, EP Rico, M de Bem Arizi, RD Dias, MR Bogo, ... Toxicology in Vitro 20 (6), 954-958, 2006 | 69 | 2006 |
Carbofuran and malathion inhibit nucleotide hydrolysis in zebrafish (Danio rerio) brain membranes MR Senger, EP Rico, M de Bem Arizi, DB Rosemberg, RD Dias, MR Bogo, ... Toxicology 212 (2-3), 107-115, 2005 | 57 | 2005 |
Schistosoma mansoni infection causes oxidative stress and alters receptor for advanced glycation endproduct (RAGE) and tau levels in multiple organs in mice RB de Oliveira, MR Senger, LM Vasques, J Gasparotto, JPA dos Santos, ... International journal for parasitology 43 (5), 371-379, 2013 | 56 | 2013 |
Kinetics Studies on the Inhibition Mechanism of Pancreatic α‐Amylase by Glycoconjugated 1H‐1,2,3‐Triazoles: A New Class of Inhibitors with Hypoglycemiant … MR Senger, LCA Gomes, SB Ferreira, CR Kaiser, VF Ferreira, FP Silva Jr ChemBioChem 13 (11), 1584-1593, 2012 | 54 | 2012 |
QSAR-Driven Discovery of Novel Chemical Scaffolds Active against Schistosoma mansoni CC Melo-Filho, RF Dantas, RC Braga, BJ Neves, MR Senger, ... Journal of chemical information and modeling 56 (7), 1357-1372, 2016 | 53 | 2016 |
COVID-19: molecular targets, drug repurposing and new avenues for drug discovery MR Senger, TCS Evangelista, RF Dantas, MVS Santana, LCS Gonçalves, ... Memórias do Instituto Oswaldo Cruz 115, e200254, 2020 | 43 | 2020 |
Kinetic characterization of adenosine deaminase activity in zebrafish (Danio rerio) brain DB Rosemberg, EP Rico, MR Senger, RD Dias, MR Bogo, CD Bonan, ... Comparative Biochemistry and Physiology Part B: Biochemistry and Molecular …, 2008 | 42 | 2008 |
Ethanol and acetaldehyde alter NTPDase and 5′-nucleotidase from zebrafish brain membranes EP Rico, DB Rosemberg, MR Senger, M de Bem Arizi, RD Dias, AA Souto, ... Neurochemistry International 52 (1-2), 290-296, 2008 | 40 | 2008 |
Acute and subchronic copper treatments alter extracellular nucleotide hydrolysis in zebrafish brain membranes DB Rosemberg, EP Rico, MR Senger, M de Bem Arizi, RD Dias, MR Bogo, ... Toxicology 236 (1-2), 132-139, 2007 | 31 | 2007 |
Design, synthesis, cholinesterase inhibition and molecular modelling study of novel tacrine hybrids with carbohydrate derivatives JPB Lopes, L Silva, G da Costa Franarin, MA Ceschi, DS Lüdtke, ... Bioorganic & medicinal chemistry 26 (20), 5566-5577, 2018 | 27 | 2018 |
Peritoneal and serum interleukin-18 levels are not increased in women with minimum or mild endometriosis C Glitz, CA Souza, GP Rodini, V Genro, JP Bilibio, M Senger, ... Brazilian Journal of Medical and Biological Research 42, 1039-1043, 2009 | 27 | 2009 |
Influence of mercury chloride on adenosine deaminase activity and gene expression in zebrafish (Danio rerio) brain MR Senger, DB Rosemberg, KJ Seibt, RD Dias, MR Bogo, CD Bonan Neurotoxicology 31 (3), 291-296, 2010 | 26 | 2010 |